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PF-06372865

Catalog No.
BA6663
PF-06372865 is an orally active, alpha2/alpha3/alpha5 subtype-selective positive alteration modulator (PAM).
Grouped product items
SizePriceStock Qty
1mL(10 mM in DMSO)
$118.00
Ship with 10-15 days
1mg
$61.00
Ship with 10-15 days
5mg
$108.00
Ship with 10-15 days
10mg
$171.00
Ship with 10-15 days
25mg
$342.00
Ship with 10-15 days
50mg
$547.00
Ship with 10-15 days
100mg
$877.00
Ship with 10-15 days
For scientific research use only and should not be used for diagnostic or medical purposes.

Tel: +1-832-696-8203

Email: [email protected]

Worldwide Distributors

Background

PF-06372865 is an orally active, α2/α3/α5 subtype-selective positive alteration modulator (PAM).PF-06372865 is a high-affinity ligand for the α1/α2/α3/α5 subunits, with values of 2.9 nM, 21 nM, and 134 nM for α2, α1PAM, and α2PAM, respectively, and low affinity for α4/α6 subunits. PF-06372865 can cross the blood-brain barrier (BBB).PF-06372865 has anxiolytic activity and has potential for use in epilepsy research.

Chemical Properties

Physical AppearanceA solid
Storage4°C, protect from light
M.Wt440.49
Cas No.1614245-70-3
FormulaC22H21FN4O3S
Shipping ConditionSmall Molecules with Blue Ice, Modified Nucleotides with Dry Ice.
General tips We do not recommend long-term storage for the solution, please use it up soon.