Histamine Receptor
Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.
- C5734 Trimipramine (maleate)Summary: potent antagonist of histamine H1 receptor
- C4255 DimebolinSummary: antihistamine, orally-available
- C4153 Doxepin (hydrochloride)Summary: histamine, serotonin, adrenergic, and muscarinic receptors antagonist
- C3989 Chlorcyclizine (hydrochloride)Summary: histamine H1 receptor antagonist and inhibits HCV
- B6156 CinnarizineSummary: antihistamine and calcium channel blocker
- B6147 CarbinoxaMine MaleateSummary: histamine-H1 receptor inhibitor
- B4843 DecloxizineSummary: histamine 1 receptor antagonist
- B5709 VUF 10460Summary: histamine H4 receptor agonist
- B5513 JNJ 5207852 dihydrochlorideSummary: histamine H3 receptor neutral antagonist
- B5021 TiotidineSummary: Potent histamine H2-receptor antagonist