HER2
- B1544 Tyrphostin AG 879Summary: HER2 inhibitor
- B1543 Mubritinib (TAK 165)Target: ErbBSummary: Potent inhibitor of HER2/ErbB2
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1) inhibitor
- A8322 Neratinib (HKI-272)3 CitationTarget: EGFRSummary: HER2/EGFR inhibitor,potent and irreversible
- A8247 Afatinib (BIBW2992)1 CitationTarget: EGFRSummary: Irreversible EGFR/HER2 inhibitor
- A8218 Lapatinib7 CitationTarget: ErbBSummary: EGFR/HER2 inhibitor,potent,selective and reversible
- A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: Multitargeted HDAC inhibitor
- A3967 Lapatinib DitosylateTarget: EGFR|ErbB-2Summary: EGFR/HER2 inhibitor,potent and selective
- A3276 Canertinib dihydrochlorideSummary: Pan-ErbB inhibitor, potent and selective
- A3252 BMS-599626 HydrochlorideSummary: EGFR/HER2 inhibitor,potent and selective