HER2
- A3145 Afatinib dimaleateTarget: EGFR|HER2Summary: EGFR inhibitor
- A2822 AC480 (BMS-599626)Target: EGFRSummary: HER1/2 inhibitor,selective and efficacious
- A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: HER2 inhibitor,potent and selective
- A1835 Pelitinib (EKB-569)Summary: EGFR inhibitor,potent and irreversible