Protein Tyrosine Kinase/RTK
-
C9130 SelitrectinibSummary: A selective TRK inhibitor, suitable for in vitro kinase signaling research, for research use only. -
C9100 Tirabrutinib HClSummary: A selective irreversible BTK inhibitor for research in immunology and tumor biology. -
C9072 DesMethyl Erlotinib HClSummary: An EGFR inhibitor compatible with CuAAC labeling, for in vitro research use. -
C8982 Pirtobrutinib (LOXO-305)Summary: A BTK inhibitor -
C8979 Pralsetinib (BLU-667)Summary: Pralsetinib (BLU-667; CAS 2097132-94-8) is a selective RET tyrosine kinase inhibitor targeting RET signaling, widely utilized in oncology and molecular signaling research. -
C8976 Avapritinib (BLU-285)Summary: Avapritinib (BLU-285; CAS 1703793-34-3) is a selective KIT and PDGFRA tyrosine kinase inhibitor widely utilized in oncology and signal transduction research. -
C8921 Ripretinib (DCC-2618)Summary: A KIT and PDGFRα inhibitor -
C8918 Ritlecitinib (PF-06651600)Summary: Ritlecitinib (PF-06651600; CAS 1792180-81-4) is a selective covalent JAK3/TEC family kinase inhibitor used to investigate cytokine signaling and immune-cell pathway biology. -
C8917 TucatinibSummary: An inhibitor of HER2 -
C8914 FursultiamineSummary: A derivative of vitamin B1

