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DiscoveryProbe™ GPCR Compound Library

Catalog No.
A unique collection of 677 GPCR-related small molecules for GPCR screening.
Grouped product items
SizePriceStock Qty
100uL/well(10 mM solution),96 Well Deep Well Plate
In stock
100uL/well(10 mM solution),96 Well Racks With Screw Cap
In stock
250uL/well(10 mM solution),96 Well Racks With Screw Cap
In stock

Tel: +1-832-696-8203

Email: [email protected]

Worldwide Distributors

Featured Products of the Library

Catalog No. Product Name Summary Targets CAS Number Smiles
A3125 5-Iodotubercidin Adenosine kinase inhibitor,potent Adenosine Kinase 24386-93-4 C1=C(C2=C(N1C3C(C(C(O3)CO)O)O)N=CN=C2N)I
A3170 AM966 LPA1 antagonist, oral active, high affinity, selective LPA Receptor 1228690-19-4 CC1=NOC(=C1NC(=O)OC(C)C2=CC=CC=C2Cl)C3=CC=C(C=C3)C4=CC=C(C=C4)CC(=O)O
A3802 SCH 527123 CXCR1 and CXCR2 receptors antagonist CXCR 473727-83-2 CCC(C1=CC=C(O1)C)NC2=C(C(=O)C2=O)NC3=CC=CC(=C3O)C(=O)N(C)C
A5827 AM1241 Cannabinoid CB2 receptor agonist,potent and selective Cannabinoid Receptor 444912-48-5 CN1CCCCC1CN2C=C(C3=CC=CC=C32)C(=O)C4=C(C=CC(=C4)[N+](=O)[O-])I
A8439 GSK1292263 Novel GPR119 agonist FFAR1 (GPR40) 1032823-75-8 CC(C)C1=NOC(=N1)N2CCC(CC2)COC3=CN=C(C=C3)C4=CC=C(C=C4)S(=O)(=O)C
B1007 AVE 0991 Agonist of angiotensin-(1-7) receptor Angiotensin Receptor 304462-19-9 CCNC(=O)NS(=O)(=O)C1=C(C=C(S1)CC(C)C)C2=CC=C(C=C2)CN3C(=C(N=C3C4=CC=CC=C4)OC)C=O
B1347 Ritodrine HCl β-2 adrenergic receptor agonist Adrenergic Receptor 23239-51-2 CC(C(C1=CC=C(C=C1)O)O)NCCC2=CC=C(C=C2)O.Cl
B1593 Irsogladine PDE4 inhibitor PDE 57381-26-7 C1=CC(=C(C=C1Cl)C2=NC(=NC(=N2)N)N)Cl
Download the GPCR-Compound-Library - XLSX       Download the GPCR-Compound-Library - SDF

Quality Control

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Clemizole hydrochloride

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Plerixafor (AMD3100)

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MK 0893

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Empagliflozin (BI 10773)

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Signaling Pathway

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Storage and Shipping Information

Form Pre-dissolved DMSO solutions Stability Solution: -20°C for 12 months, -80°C for 24 months
Packaging 96-well rack with Matrix 2D Barcoded ScrewTop Storage tubes (250 μL or 100 μL/well, 10 mM DMSO).
96-well DeepWell format with peelable foil seal and EVA cap (100 μL/well, 10 mM DMSO).
General tips For obtaining a higher solubility, please warm the tube at 37°C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20°C for several months.
Shipping Condition Evaluation sample solution: ship with blue ice
All other available size: ship with RT, or blue ice upon request

Compound Library Composition


Available in stock with overnight delivery and free shipping over $500 Cost-effective and competitive price to save your findings Potent, selective and cell-permeable in inhibiting or activating target molecules Diverse in chemical structure and route of administration (oral/i.m/i.v injection etc.) Detailed files describing potency, selectivity and applications etc. Supported by published data from top peer-reviewed journals Guaranteed high quality with NMR and HPLC validation