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Apoptosis/Autophagy

Items 1-10 of 17

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  1. Pexidartinib (PLX3397)
    B5854 Pexidartinib (PLX3397)
     3 Citation
    Target: FLT3|c-Kit|CSF1R
    Summary: A multi-targeted receptor tyrosine kinase inhibitor; A CSF-1R inhibitor
      insoluble in EtOH; insoluble in H2O; ≥20.9 mg/mL
  2. Zebularine
    A1915 Zebularine
     1 Citation
    Target: DNA Methyltransferases|Cytidine deaminases
    Summary: Cytidine analog; DNA methyltransferase (DNMT) inhibitor; induces DNA demethylation
      insoluble in EtOH; ≥50.7 mg/mL
  3. Valproic acid sodium salt
    A4099 Valproic acid sodium salt
    Target: Histone Deacetylases (HDACs)
    Summary: A class I HDAC inhibitor
      ≥8.35 mg/mL
  4. U0126
    BA2003 U0126
    Summary: A potent, non-ATP-competitive, selective MEK inhibitor
      ≥23.15 mg/mL
  5. PD 173074
    A8253 PD 173074
     5 Citation
    Target: VEGFR|FGFR
    Summary: FGFR inhibitor
      ≥26.18 mg/mL
  6. Curcumin
    A3335 Curcumin
     1 Citation
    Target: Histone Deacetylases (HDACs)|Nrf2|Histone Acetyltransferases (HATs)|Tyrosinases
    Summary: Specific histone and non-histone acetyltransferase inhibitor
      ≥36.8 mg/mL
  7. Telaglenastat
    B4799 Telaglenastat
     1 Citation
    Target: Glutaminases
    Summary: Orally active glutaminase inhibitor
      ≥28.6 mg/mL
  8. Dextran sulfate sodium salt (MW 35000-45000)
    B8205 Dextran sulfate sodium salt (MW 35000-45000)
    Summary: Nucleic acid hybridization enhancer; for acute or chronic colitis models
      insoluble in EtOH; insoluble in DMSO; ≥55.5 mg/mL
  9. Lithocholic Acid
    A8463 Lithocholic Acid
    Target: Farnesoid X receptors (FXRs)|Vitamin D receptors (VDRs)|Pregnane X receptor(PXR)
    Summary: Toxic secondary bile acid; induces intrahepatic cholestasis; FXR antagonist and PXR/SXR agonist
      insoluble in H2O; ≥12.95 mg/mL
  10. Tamoxifen
    B5965 Tamoxifen
     17 Citation
    Target: PKC
    Summary: estrogen receptor modulator
      ≥18.6 mg/mL

Items 1-10 of 17

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