TGF-βR1(ALK5)
TGF-βR1 (transforming growth factor beta receptors) are a serine/threonine protein kinase that involved in the regulation of cell cycle arrest, cell proliferation and differentiation, production of extracellular matrix, wound healing, tumorgenesis and immunosuppression etc.
- A3132 A 77-01Summary: Potent ALK5 inhibitor
- A3133 A 83-01Summary: ALK inhibitor
- A3799 SB-505124 hydrochlorideTarget: ALKSummary: ALK5/ALK4/ALK7 inhibitor in TGF-β/activin signalling,selective
- A3808 SD-208Summary: TGF-βR I kinase inhibitor
- A5602 SB525334Summary: (TGF-beta1) receptor inhibitor
- A8301 GW788388Summary: ALK5 inhibitor, potent and selective
- A8348 LY21572992 CitationSummary: TGF-βR1 inhibitor,potent and selective
- A8464 LY21097614 CitationSummary: TβRI/II kinase inhibitor
- B2286 K02288Target: ALKSummary: ALK inhibitor
- C3656 ALK5 Inhibitor II (hydrochloride)Summary: ALK5 inhibitor