TRPV1
TRPV1 (transient receptor potential vanilloid 1) is a calcium permeant cation channel that detects thermal stimuli and noxious chemical. It is a drug target for analgesics.
- A1174 AMG-517Target: TRP ChannelSummary: TRPV1 antagonist,potent and highly selective
- A8519 SB705498Summary: TRPV1 antagonist,potent and selective
- B5930 mavatrepSummary: TRPV1 antagonist
- C4082 Eicosapentaenoyl SerotoninSummary: TRPV1 channel inhibitor
- C4167 Oleoyl SerotoninSummary: TRPV1 channel inhibitor
- C4169 Palmitoyl SerotoninSummary: TRPV1 channel inhibitor
- C4170 Stearoyl SerotoninSummary: TRPV1 channel inhibitor
- C4171 Docosahexaenoyl SerotoninSummary: TRPV1 channel inhibitor
- C4563 CapsiconiateSummary: TRPV1 agonist
- A3279 CapsazepineSummary: TRPV1 ion channel antagonist