Endothelin Receptor
Endothelin receptors are members of rhodopsin-like g-protein coupled receptor (GPCRA) with 4 types (ETA, ETB1, ETB2 and ETC), which mediate various physiological processes including vasoconstriction, vasodilation, and neurotransmission etc.
- A5489 Zibotentan (ZD4054)1 CitationSummary: ETA receptor antagonist,potent and specific
- A1929 MacitentanSummary: Endothelin (ET)(A) and ET(B) receptor antagonist
- B1682 BosentanSummary: Endothelin receptor antagonist
- B1521 Bosentan HydrateSummary: endothelin receptor antagonist
- B5062 Endothelin 3 (human, rat)Summary: Endogenous neuropeptide with selectivity for the putative ETC endothelin receptor
- B5069 Sarafotoxin S6bSummary: non-selective endothelin receptor agonist
- B5217 Sarafotoxin S6aSummary: Endothelin receptor agonist
- A3201 Atrasentan hydrochlorideSummary: Endothelin receptor antagonist
- A3208 AvosentanSummary: ETA receptor antagonist