CFTR
CFTR (cystic fibrosis transmembrane conductance regulator) is an ABC transporter-class ion channel that conducts chloride[3] and thiocyanate[4] ions across epithelial cell membranes.
- B1087 GlyH-101Target: CFTRSummary: CFTR Inhibitor II
- B1435 CFTRinh-172Summary: CFTR inhibitor, highly potent and selective
- B3504 PPQ-102Summary: potent CFTR inhibitor
- A3510 Ivacaftor benzenesulfonateSummary: CFTR Potentiator
- A3511 Ivacaftor hydrateSummary: CFTR Potentiator
- A5047 Ivacaftor (VX-770)1 CitationSummary: Potent CFTR potentiator
- A2664 VX-661Target: CFTRSummary: F508del CFTR corrector
- A8351 VX-809Target: CFTRSummary: CFTR corrector
- A8553 PTC124 (Ataluren)Summary: CFTR-G542X nonsense allele inhibitor
- A8637 IOWH-032Target: CFTRSummary: CFTR inhibitor