Adrenergic Receptor
Adrenergic receptor is a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.
- C5822 p-iodo-Clonidine (hydrochloride)Summary: partial agonist of the α2-adrenergic receptor
- C5802 CarazololSummary: high-affinity, lipophilic, non-selective ligand of the β-adrenergic receptors
- C5675 Fendiline (hydrochloride)Summary: α2-adrenergic receptor antagonist
- C5580 AnisodamineSummary: weak antagonist of α1-adrenoceptors
- C5286 (R,S)-AtenololSummary: β1-adrenergic receptor antagonist
- C5043 Bufuralol (hydrochloride)Summary: non-specific β-adrenergic blocker
- C4521 Celiprolol (hydrochloride)Summary: β1 adrenergic receptor antagonist and β2 adrenergic receptor partial agonist
- C3031 (R)-(+)-AtenololSummary: less active enantiomer of the racemic β1-adrenergic receptor antagonist, (R,S)-atenolol.
- C3003 (±)-TalinololSummary: β1-selective adrenoceptor antagonist
- C4493 Midodrine (hydrochloride)Summary: prodrug of the α1-adrenergic receptor agonist