MEK1/2
MEK1/2, also known as MAPKK (mitogen-activated protein kinase kinase), is a kinase enzyme which phosphorylates MAPK (mitogen-activated protein kinase).
- A8207 AZD6244 (Selumetinib)3 CitationSummary: MEK inhibitor
- A1663 PD980599 CitationTarget: MEKSummary: MEK inhibitor,selective and reversible
- A1894 SL-3271 CitationTarget: MEKSummary: Selective MEK1/2 inhibitor
- A1792 PD184352 (CI-1040)Target: MEKSummary: Selective MEK inhibitor
- A1337 U0126-EtOH10 CitationTarget: MEKSummary: MEK1/2 inhibitor
- A5573 Pimasertib (AS-703026)Target: MEKSummary: MEK1/2 inhibitor
- A5707 PD318088Target: MEKSummary: Allosteric MEK1/2 inhibitor, non-ATP competitive
- A5801 BIX 02189Target: MEK|ERKSummary: Selective MEK5 inhibitor
- A5803 BIX 02188Target: MEKSummary: MEK5 inhibitor,potent and selective
- A1947 MEK162 (ARRY-162, ARRY-438162)Target: MEKSummary: MEK1/2 inhibitor,potent and selective