EZH2
EZH2 (enhancer of zeste homolog 2) is a polycomb group protein and histone methyltrasferase that associated with transcriptional repression. It catalyzes trimethylation of H3K27me3 (histone H3 lysine 27) as a catalytic subunit of PRC2 (polycomb repressive complex 2).
- 2 CitationSummary: EZH2 inhibitor
- 1 CitationTarget: EZH2|EZH1Summary: EZH2 inhibitor
- Summary: EZH2 inhibitor
- 1 CitationTarget: EZH2Summary: EZH2 inhibitor,potent,selective and cell permeable
- 5 CitationTarget: EZH2Summary: EZH2 inhibitor
- 6 CitationTarget: HydrolaseSummary: S-adenosylhomocysteine and EZH2 inhibitor
- 2 CitationTarget: EZH2Summary: EZH2 inhibitor,potent and selective
- 1 CitationTarget: EZH2Summary: SAHH and EZH2 inhibitor