EZH2
EZH2 (enhancer of zeste homolog 2) is a polycomb group protein and histone methyltrasferase that associated with transcriptional repression. It catalyzes trimethylation of H3K27me3 (histone H3 lysine 27) as a catalytic subunit of PRC2 (polycomb repressive complex 2).
- B5833 GSK5032 CitationSummary: EZH2 inhibitor
- A4171 EPZ0056872 CitationTarget: EZH2Summary: EZH2 inhibitor,potent and selective
- A1905 3-Deazaneplanocin,DZNep6 CitationTarget: HydrolaseSummary: S-adenosylhomocysteine and EZH2 inhibitor
- A3446 GSK1265 CitationTarget: EZH2Summary: EZH2 inhibitor
- A3449 GSK3431 CitationTarget: EZH2Summary: EZH2 inhibitor,potent,selective and cell permeable
- B1021 EI1Summary: EZH2 inhibitor
- A8182 3-Deazaneplanocin A (DZNep) hydrochloride1 CitationTarget: EZH2Summary: SAHH and EZH2 inhibitor
- B4678 CPI-1691 CitationTarget: EZH2|EZH1Summary: EZH2 inhibitor