RARs
RARs (retinoic acid receptors) are type of nuclear receptors which also act as transcription factors that are activated by both all-trans retinoic acid and 9-cis retinoic acid.
- A5710 TazaroteneSummary: Topical retinoid;antiproliferative;inducer of TIG3 tumor suppressor
- A8539 Tretinoin (Aberela)Target: RAR/RXRSummary: retinoic acid, treats acne vulgaris and keratosis pilaris
- B5438 BMS 753Summary: RARα-selective agonist
- B5483 CD 2314Summary: RARβ agonist,potent and selective
- C5100 LuffariellolideSummary: agonist for the RA receptors RAR α, β, and γ
- B2058 TTNPB (Arotinoid Acid)1 CitationTarget: RARsSummary: Potent RAR agonist
- B7396 BMS 453Summary: RAR agonist
- B6785 CD 437Target: RAR/RXRSummary: RARγ-selective agonist,potent and cell-permeable
- B6927 Ch 55Summary: RAR agonist
- B6928 LE 135Summary: RARβ antagonist