PDE
PDE (phosphodiesterases) catalyze the hydrolysis of cGMP and/or cAMP. Stimulus such as light, neurotransmitter and hormone trigger PDE to regulate various biological response including vascular smooth muscle proliferation/contraction, hormone secretion and plate aggregation etc.
- B5162 T 0156 hydrochlorideSummary: inhibitor of phosphodiesterase type 5 (PDE5)
- B5630 PiclamilastSummary: PDE4 inhibitor
- B5642 TC-E 5005Summary: PDE10A inhibitor
- B6073 Sildenafil mesylateSummary: PDE5 inhibitor
- C3266 Amino TadalafilSummary: analog of tadalafil, a potent inhibitor of phosphodiesterase 5
- C3510 MBCQSummary: cGMP-specific phosphodiesterase PDE V inhibitor
- C4796 EggmanoneSummary: selective inhibitor of PDE4
- C4686 2-Acetamidophenyl 5-chloro-2-nitrophenyl sulfideSummary: phosphodiesterase 7 (PDE7) inhibitor
- C4805 ML-030Summary: PDE4 inhibitor
- C4942 Sp-Cyclic AMPS (sodium salt)Summary: cAMP derivative used to bind PDE10 GAF domain