Muscarinic Receptor
Muscarinic receptor is a group of G-protein coupled receptors that binds to acetylcholine and mediates cellular responses, including inhibition of acetylate cyclase, phosphoinositide degradation and regulation of potassium channels. It is involved in the neurological diseases such as Alzheimer's and Parkinson's.
- B1598 Biperiden HCl1 CitationTarget: M1 ReceptorsSummary: Anticholinergic drug
- B5579 VU 0365114Summary: positive allosteric modulator of M5
- B5632 PTAC oxalateSummary: muscarinic receptor ligand
- B1609 Aclidinium BromideSummary: LAMAs antagonist
- B1620 Tolterodine tartrateTarget: AChRSummary: Competitive muscarinic receptor antagonist
- B1614 Solifenacin succinateTarget: M3 ReceptorsSummary: Muscarinic receptor antagonist
- B1600 Darifenacin HBrTarget: M3 ReceptorsSummary: Selective M3 muscarinic receptor antagonist
- B1618 Fesoterodine FumarateSummary: Muscarinic AChR receptor antagonist
- B6130 Trihexyphenidyl hydrochlorideSummary: antiparkinsonian agent of the antimuscarinic class
- C3017 Guvacoline (hydrobromide)Summary: full agonist of atrial and ileal muscarinic receptors