Muscarinic Receptor
Muscarinic receptor is a group of G-protein coupled receptors that binds to acetylcholine and mediates cellular responses, including inhibition of acetylate cyclase, phosphoinositide degradation and regulation of potassium channels. It is involved in the neurological diseases such as Alzheimer's and Parkinson's.
- B5579 VU 0365114Summary: positive allosteric modulator of M5
- B5632 PTAC oxalateSummary: muscarinic receptor ligand
- A3299 CevimelineSummary: Muscarinic receptor agonist
- A3300 Cevimeline hydrochloride hemihydrateSummary: Agonist of muscarinic receptor (M1/M3)
- B6130 Trihexyphenidyl hydrochlorideSummary: antiparkinsonian agent of the antimuscarinic class
- C3017 Guvacoline (hydrobromide)Summary: full agonist of atrial and ileal muscarinic receptors
- C3869 BQCATarget: AChRSummary: positive allosteric modulator of the M1 muscarinic acetylcholine receptor (mAChR)
- C4093 N-IsopropylnoratropineSummary: used in the synthesis of ipratropium, a muscarinic antagonist
- C4635 Aceclidine (hydrochloride)Summary: agonist of muscarinic receptors
- B1609 Aclidinium BromideSummary: LAMAs antagonist