FLT3
FLT3 (FMS-like tyrosine kinase 3) is a cytokine receptor which belongs to the receptor tyrosine kinase class III and plays a role in cell survival, proliferation, and differentiation.
- A4513 Lestaurtinib1 CitationSummary: JAK2/FLT3/TrkA inhibitor
- A2949 Linifanib (ABT-869)Target: VEGFR|PDGFRSummary: VEGFR/PDGFR inhibitor
- A2977 Cabozantinib (XL184, BMS-907351)Summary: VEGFR2/Met/Ret/Kit/FLT//AXL inhibitor
- A5467 Ponatinib (AP24534)1 CitationTarget: VEGFR|PDGFR|Bcr-Abl|FGFR|SrcSummary: pan-BCR-ABL inhibitor,multi-kinase inhibitor
- A5793 Quizartinib (AC220)Target: FLT3Summary: FLT3 inhibitor,potent and selective
- A2323 TCS 359Summary: Potent FLT3 inhibitor
- B1526 Tandutinib (MLN518)Summary: FLT3 inhibitor,potent and selective
- B5516 5'-FluoroindirubinoximeSummary: FMS-like receptor tyrosine kinase-3 (FLT3) inhibitor
- A8889 G-749Target: Aurora Kinases|FLT3|c-RETSummary: FLT3 inhibitor
- B8016 UNC20251 CitationTarget: MER|FLT3Summary: orally bioavailable dual MER/FLT3 inhibitor