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DiscoveryProbe™ Tyrosine Kinase Inhibitor Library
A unique collection of 247 tyrosine kinase inhibitors for high throughput screening (HTS) and high content screening (HCS).

DiscoveryProbe™ Tyrosine Kinase Inhibitor Library

Catalog No. L1028
Size Price Stock Qty
100uL/well(10 mM solution) $4,220.00 In stock
250uL/well(10 mM solution) $7,530.00 In stock
5mg/well $9,840.00 In stock

Tel: +1-832-696-8203

Email: sales@apexbt.com

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Sample solution is provided at 25 µL, 10mM.

Click and Customize the Panel with your own choices of compounds/size/quantities/chemical forms etc.

HTS Facility Partners

Featured Products of the Library

Catalog No. Product Name Summary Targets CAS Number Smiles
A1389 WZ4002 Mutant-selective EGFR inhibitor(L858R,T790M), irreversible and potent EGFR 1213269-23-8 CN1CCN(CC1)C2=CC(=C(C=C2)NC3=NC=C(C(=N3)OC4=CC=CC(=C4)NC(=O)C=C)Cl)OC
A2838 OSI-930 Inhibitor of Kit, KDR, Flt, CSF-1R, c-Raf and Lck c-Kit 728033-96-3 C1=CC=C2C(=C1)C(=CC=N2)CNC3=C(SC=C3)C(=O)NC4=CC=C(C=C4)OC(F)(F)F
A3014 BGJ398 FGFR inhibitor ,potent and selective FGFR 872511-34-7 CCN1CCN(CC1)C2=CC=C(C=C2)NC3=CC(=NC=N3)N(C)C(=O)NC4=C(C(=CC(=C4Cl)OC)OC)Cl
A5092 JNJ-38877605 C-Met inhibitor,ATP-competitive c-MET 943540-75-8 CN1C=C(C=N1)C2=NN3C(=NN=C3C(C4=CC5=C(C=C4)N=CC=C5)(F)F)C=C2
A8324 LDN-193189 ALK inhibitor,potent and selective SMAD 1062368-24-4 C1CN(CCN1)C2=CC=C(C=C2)C3=CN4C(=C(C=N4)C5=CC=NC6=CC=CC=C56)N=C3
A8329 R428 Selective Axl inhibitor Axl 1037624-75-1 C1CCN(C1)C2CCC3=C(CC2)C=C(C=C3)NC4=NN(C(=N4)N)C5=NN=C6C(=C5)CCCC7=CC=CC=C76
A8528 TAK-285 HER2/EGFR(HER1) inhibitor HER2 871026-44-7 CC(C)(CC(=O)NCCN1C=CC2=C1C(=NC=N2)NC3=CC(=C(C=C3)OC4=CC=CC(=C4)C(F)(F)F)Cl)O
A8696 FIIN-2 Irreversible inhibitor of FGFR EGFR 1633044-56-0 O=C(C=C)NC1=CC=C(CN2C(N(C3=CC(OC)=CC(OC)=C3)CC4=CN=C(NC5=CC=C(N6CCN(C)CC6)C=C5)N=C42)=O)C=C1
Download the Tyrosine-Kinase-Inhibitor-Library - XLSX       Download the Tyrosine-Kinase-Inhibitor-Library - SDF

Quality Control

Related Biological Data

GSK1904529A

Related Biological Data

GSK1904529A

Related Biological Data

R428

Related Biological Data

R428

Related Biological Data

Bafetinib

Signaling Pathway

Bcr-Abl Compare Products
PKC Compare Products
ROCK Compare Products

Advantages

  • Available in stock with overnight delivery and free shipping over $500
  • Cost-effective and competitive price to save your findings
  • Potent, selective and cell-permeable in inhibiting or activating target molecules
  • Diverse in chemical structure and route of administration (oral/i.m/i.v injection etc.)
  • Detailed files describing potency, selectivity and applications etc.
  • Supported by published data from top peer-reviewed journals
  • Guaranteed high quality with NMR and HPLC validation

Storage and Shipping Information

Form Pre-dissolved DMSO solutions Stability -20°C: 12 months
-80°C: 24 months
Packaging 96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode.
General tips For obtaining a higher solubility , please warm the tube at 37°C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20°C for several months.
Shipping Condition Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request

Compound Library Composition