PI3K
PI3K (phosphatidylinositol-4,5-bisphosphate 3-kinase) is a family of enzymes involved in cellular functions such as cell growth, proliferation, differentiation, motility, survival and intracellular trafficking, which in turn are involved in cancer.
- N1841 QuercetinSummary: Antitumor agent
- B2180 AS-252424Target: Akt|PI3KSummary: PI3Kγ inhibitor,novel and potent
- B2181 AS-604850Summary: PI3Kγ inhibitor,selective and ATP-competitve
- B2187 PIK-293Summary: PI3K inhibitor
- B2188 PIK-294Summary: highly selective p110δ inhibitor
- B2177 TG100713Target: PI3KSummary: pan-PI3K inhibitor
- B2182 CAY10505Summary: Potent PI3Kγ inhibitor
- B4660 PI-3065Target: PI3KSummary: P110δkinase inhibitor
- A4097 CUDC-907Target: Histone Deacetylases (HDACs)|PI3KSummary: Potent PI3K/HDAC inhibitor
- A3238 BEZ235 Tosylate1 CitationSummary: MTOR/P13K inhibitor