PI3K
PI3K (phosphatidylinositol-4,5-bisphosphate 3-kinase) is a family of enzymes involved in cellular functions such as cell growth, proliferation, differentiation, motility, survival and intracellular trafficking, which in turn are involved in cancer.
- A8210 GDC-094110 CitationTarget: PI3KSummary: PI3K inhibitor,potent and selective
- A8246 BEZ235 (NVP-BEZ235)2 CitationSummary: PI3K/mTOR inhibitor,ATP-competitve
- A8248 ZSTK474Summary: Potent PI3K inhibitor
- A8250 LY 29400216 CitationTarget: PI3KSummary: Potent PI3K inhibitor
- A2067 PI-1031 CitationSummary: Class I PI3K, mTOR and DNA-PK inhibitor
- A5112 XL147Target: PI3KSummary: PI3K inhibitor,selective and reversible
- A2681 TGX-221Target: PI3KSummary: PI3Kβ inhibitor,potent,selective and ATP competitive
- A2552 Quercetin dihydrateTarget: PI3K|PIM1 kinase|phospholipase A2Summary: PLA2 and PI 3-kinase inhibitor
- A2754 TG100-115Target: PI3KSummary: PI3Kγ/PI3Kδ inhibitor
- A2764 PIK-90Summary: PI3K inhibitor,potent selective