P-gp
P-gp (P-glycoprotein) is a ATP-binding cassette transproters which overepxressed in multidrug-resistance cancer cells. It functions in pumping drug out of cell and lower intracellular drug concentration.
- A8549 LY335979 (Zosuquidar 3HCL)1 CitationTarget: P-glycoprotein (P-gp)Summary: Pgp (P-glycoprotein) inhibitor
- C3140 Rhodamine 123 (chloride)Summary: membrane-permeable cationic dye used as substrate for the efflux pump P-glycoprotein
- C3610 HypophyllanthinSummary: P-glycoprotein (P-gp) inhibitor
- C3897 Estradiol 3-(β-D-Glucuronide) (sodium salt)Summary: substrate for multidrug resistance protein 2 (MRP2)
- C3840 Estradiol 17-(β-D-Glucuronide) (sodium salt)Summary: substrate of the multidrug resistance protein 2 (MRP2)
- B1167 Dofequidar fumarateSummary: MDR reversal agent
- A8208 Tariquidar2 CitationTarget: P-glycoprotein (P-gp)Summary: P-glycoprotein inhibitor,potent and non-competitive
- A3859 Tariquidar methanesulfonate, hydrateTarget: P-glycoprotein (P-gp)Summary: P-glycoprotein inhibitor, potent and selective
- A3956 ZosuquidarTarget: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)Summary: MDR modulator