Androgen Receptor
AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.
- B5481 TFM-4AS-1Summary: androgen receptor modulator
- A8452 ODM-201Target: Androgen ReceptorsSummary: new-generation androgen receptor inhibitor
- B6041 EPI-001Summary: AR antagonist
- C3186 RD162Summary: androgen receptor (AR) antagonist
- C3546 HE-3235Summary: androgen receptor antagonist
- C3644 DanazolSummary: weak androgenic effects
- C4317 5α-dihydro-11-keto TestosteroneSummary: androgen receptor agonist
- C4721 2-hydroxy FlutamideSummary: androgen receptor inhibitor
- C4768 GSK2881078Summary: selective androgen receptor modulator (SARM)
- A3003 MDV3100 (Enzalutamide)12 CitationTarget: Androgen ReceptorsSummary: Androgen receptor antagonist