Rho
Rho GTPases act as molecular switches that convert and amplify external signals into cellular effects upon activation of cell surface receptor in various signaling transduction pathway. It functions in cell proliferation, motility, survival cytoskeletal remodeling and membrane trafficking etc.
- A1352 Zoledronic AcidTarget: Farnesyl Diphosphate SynthasesSummary: Potent nitrogen-containing bisphosphonates
- A1952 NSC23766 trihydrochlorideSummary: Selective inhibitor of Rac1-GEF interaction.
- A8300 ZCL2781 CitationTarget: Cdc42Summary: Selective Cdc42 inhibitor
- C5799 (R)-CCG-1423Summary: Rho inhibitor
- C5803 (S)-CCG-1423Summary: Rho inhibitor
- B5529 SB 772077B dihydrochlorideSummary: Rho-kinase (ROCK) inhibitor
- B5773 AS 1892802Summary: ROCK inhibitor,potent and ATP-competitive
- A8902 6H05Summary: K-Ras inhibitor
- B4809 K-115Summary: Selective Rho kinase inhibitor
- B4897 CCG-1423Target: RhoSummary: RhoA inhibitor