ATM/ATR
ATM (ataxia telangiectasia mutated) and ATR (ATM- and Rad3-related) are two PIKKs (phosphatidylinositol 3-kinase-like kinases) that regulate the DNA damage response (DDR) pathways.
- A4605 KU 559331 CitationSummary: ATM inhibitor,potent and selective
- A2521 VE-8212 CitationSummary: ATR kinase inhibitor
- A8336 KU-600192 CitationTarget: ATM/ATRSummary: ATM kinase inhibitor,potent and selective
- A8624 CGK733Target: ATM/ATRSummary: ATM/ATR inhibitor,potent and selective
- A8625 CP-466722Target: ATMSummary: ATM inhibitor,potent and reversible
- A8626 ETP-46464Target: PI3K|mTOR|DNA-PK|ATM/ATRSummary: ATR inhibitor,potent and selective
- B1383 VE-8222 CitationTarget: ATM/ATRSummary: ATR inhibitor
- B5389 MirinSummary: A potent inhibitor of the Mre11-Rad50-Nbs1 (MRN)-ATM pathway
- A3210 AZ201 CitationTarget: ATM/ATRSummary: ATR inhibitor,potent and selective