EGFR
EGFR (epidermal growth factor receptor) is the cell-surface receptor of its specific ligands, including epidermal growth factor and TGFα (transforming growth factor α) and is a receptor tyrosine kinase.
- B5836 AZ5104Target: EGFRSummary: EGFR inhibitor
- B5962 AZD3759Summary: EGFR inhibitor,oral active
- B6115 RG 13022Summary: EGFR tyrosine kinase inhibitor
- B1103 Mutant EGFR inhibitorSummary: Selective Mutated EGFR inhibitor
- B1496 IcotinibSummary: EGFR tyrosine kinase inhibitor
- B1104 AZD-92911 CitationTarget: EGFRSummary: Mutated forms EGFR inhibitor
- B1105 AZD-9291 mesylateSummary: third generation EGFRm inhibitor, oral and irreversible
- A8319 Dacomitinib (PF299804, PF299)Target: ErbBSummary: HER inhibitor
- A8322 Neratinib (HKI-272)1 CitationTarget: EGFRSummary: HER2/EGFR inhibitor,potent and irreversible
- A8357 AG-1478Target: EGFRSummary: EGFR inhibitor,potent and selective