CCR2
CCR2 (C-C chemokine receptor type 2), the receptor for monocyte chemoattractant protein-1 (CCL2), mediate agonist-dependent calcium mobilization and inhibition of adenylyl cyclase.
- A3492 INCB 3284 dimesylateSummary: HCCR2 antagonist
- A3494 INCB3344Target: CCRSummary: CCR2 chemokine receptor antagonist
- A3495 INCB8761(PF-4136309)Summary: CCR2 Antagonist,potent and selective
- A3611 MK-0812Summary: antagonist of chemokine receptor CCR-2
- A3779 RS 5043931 CitationSummary: CCR2 chemokine receptor antagonist