Anti-infection
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BA1942 Darunavir-d9Summary: Darunavir-d9 (TMC114-d9) is the deuterium substitute for Darunavir. -
BA1943 NifevirocSummary: Nifeviroc is an antagonist with oral activity. -
BA1948 2-Deoxy-2-fluoroarabinoadenosineSummary: 2'-Deoxy-2'-fluoroarabinoadenosine is a nucleoside analog. -
BA1951 DPC-681Summary: DPC-681 is a potent and selective HIVprotease inhibitor. -
BA1953 PirmitegravirSummary: Pirmitegravir is a potent, first-in-class inhibitor targeting the LEDGF/p75 binding site. -
BA1958 PeldesineSummary: Peldesine (BCX34) is a potent, competitive, reversible and orally active purine nucleoside phosphorylase inhibitor. -
BA1959 AzddMeCSummary: AzddMeC (CS-92) is an antiviral nucleoside analog and a potent, selective, orally active inhibitor of reverse transcriptase and replication. -
BA1966 BDM-2Summary: BDM-2 is an IN-LEDGF-altering inhibitor (INLAI) of integrase (=47nM) and has potent antiretroviral (ARV) activity. -
BA1976 HIV-IN-6Summary: HIV-IN-6 is an HIV-I viral replication inhibitor. -
BA1977 CDK9-IN-30Summary: CDK9-IN-30 is an inhibitor.
