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MK-2461

MK-2461

Catalog No. A8476
Size Price Stock Qty
5mg $284.00 In stock
10mg $498.00 In stock

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Sample solution is provided at 25 µL, 10mM.

MK-2461 Dilution Calculator

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MK-2461 Molarity Calculator

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Chemical Properties

Cas No. 917879-39-1 SDF Download SDF
Chemical Name 9-[[[(2R)-1,4-dioxan-2-yl]methyl-methylsulfamoyl]amino]-2-(1-methylpyrazol-4-yl)-11-oxobenzo[1,2]cyclohepta[2,4-b]pyridine
Canonical SMILES CN1C=C(C=N1)C2=CN=C3C=CC4=C(C=C(C=C4)NS(=O)(=O)N(C)CC5COCCO5)C(=O)C3=C2
Formula C24H25N5O5S M.Wt 495.55
Solubility Soluble in DMSO Storage Store at -20°C
Shipping Condition: Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request

Background

MK-2461 is a potent inhibitor of Met, Ron, Flt1, Flt 3, PDGFRβ, and Mer with IC50 of 2.5 nM, 7 nM, 10 nM, 22 nM, 22 nM and 24 nM, respectively.