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DiscoveryProbe™ GPCR Compound Library
A unique collection of 528 GPCR-related small molecules for GPCR screening.

Catalog No.L1025
Size Price Stock Qty
100uL/well(10 mM solution)
$4,040.00
In stock
250uL/well(10 mM solution)
$7,300.00
In stock
5mg/well
$9,500.00
In stock

Tel: +1-832-696-8203

Email: [email protected]

Worldwide Distributors

      

Sample solution is provided at 25 µL, 10mM.

Click and Customize the Panel with your own choices of compounds/size/quantities/chemical forms etc.

HTS Facility Partners

HTS Facility Partners

Featured Products of the Library

Catalog No. Product Name Summary Targets CAS Number Smiles
A3125 5-Iodotubercidin Adenosine kinase inhibitor,potent Adenosine Kinase 24386-93-4 C1=C(C2=C(N1C3C(C(C(O3)CO)O)O)N=CN=C2N)I
A3170 AM966 LPA1 antagonist, oral active, high affinity, selective LPA Receptor 1228690-19-4 CC1=NOC(=C1NC(=O)OC(C)C2=CC=CC=C2Cl)C3=CC=C(C=C3)C4=CC=C(C=C4)CC(=O)O
A3802 SCH 527123 CXCR1 and CXCR2 receptors antagonist CXCR 473727-83-2 CCC(C1=CC=C(O1)C)NC2=C(C(=O)C2=O)NC3=CC=CC(=C3O)C(=O)N(C)C
A5827 AM1241 Cannabinoid CB2 receptor agonist,potent and selective Cannabinoid Receptor 444912-48-5 CN1CCCCC1CN2C=C(C3=CC=CC=C32)C(=O)C4=C(C=CC(=C4)[N+](=O)[O-])I
A8439 GSK1292263 Novel GPR119 agonist FFAR1 (GPR40) 1032823-75-8 CC(C)C1=NOC(=N1)N2CCC(CC2)COC3=CN=C(C=C3)C4=CC=C(C=C4)S(=O)(=O)C
B1007 AVE 0991 Agonist of angiotensin-(1-7) receptor Angiotensin Receptor 304462-19-9 CCNC(=O)NS(=O)(=O)C1=C(C=C(S1)CC(C)C)C2=CC=C(C=C2)CN3C(=C(N=C3C4=CC=CC=C4)OC)C=O
B1347 Ritodrine HCl β-2 adrenergic receptor agonist Adrenergic Receptor 23239-51-2 CC(C(C1=CC=C(C=C1)O)O)NCCC2=CC=C(C=C2)O.Cl
B1593 Irsogladine PDE4 inhibitor PDE 57381-26-7 C1=CC(=C(C=C1Cl)C2=NC(=NC(=N2)N)N)Cl
Download the GPCR-Compound-Library - XLSX       Download the GPCR-Compound-Library - SDF

Quality Control

Related Biological Data

Clemizole hydrochloride

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Plerixafor (AMD3100)

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MK 0893

Related Biological Data

Empagliflozin (BI 10773)

Related Biological Data

Dapagliflozin

Related Biological Data

Dapagliflozin

Signaling Pathway

Dehydrogenase Compare Products
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Advantages

  • Available in stock with overnight delivery and free shipping over $500
  • Cost-effective and competitive price to save your findings
  • Potent, selective and cell-permeable in inhibiting or activating target molecules
  • Diverse in chemical structure and route of administration (oral/i.m/i.v injection etc.)
  • Detailed files describing potency, selectivity and applications etc.
  • Supported by published data from top peer-reviewed journals
  • Guaranteed high quality with NMR and HPLC validation

Storage and Shipping Information

Form Pre-dissolved DMSO solutions Stability -20°C: 12 months
-80°C: 24 months
Packaging 96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode.
General tips For obtaining a higher solubility , please warm the tube at 37°C and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20°C for several months.
Shipping Condition Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request

Compound Library Composition