MEK1/2
- B5126 10Z-HymenialdisineSummary: Pan kinase inhibitor
- B3261 RO4987655Summary: MEK inhibitor
- B1621 TAK-733Target: MEKSummary: MEK allosteric site inhibitor
- B1267 RefametinibTarget: MEKSummary: MEK 1/ MEK 2 inhibitor
- B1135 GDC-0623Target: MEKSummary: MEK1 inhibitor, potent and ATP-uncompetitive
- A9907 MEK Inhibitor SetSummary: For phosphorylation and dephosphorylation applications
- A8374 AZD8330Target: MEKSummary: MEK 1/2 inhibitor
- A8207 AZD6244 (Selumetinib)3 CitationSummary: MEK inhibitor
- A5803 BIX 02188Target: MEKSummary: MEK5 inhibitor,potent and selective
- A5801 BIX 02189Target: MEK|ERKSummary: Selective MEK5 inhibitor