PI3K
PI3K (phosphatidylinositol-4,5-bisphosphate 3-kinase) is a family of enzymes involved in cellular functions such as cell growth, proliferation, differentiation, motility, survival and intracellular trafficking, which in turn are involved in cancer.
- B2182 CAY10505Summary: Potent PI3Kγ inhibitor
- B4660 PI-3065Target: PI3KSummary: P110δkinase inhibitor
- B5246 740 Y-P19 CitationTarget: PI3KSummary: PI 3-kinase activator,cell permeable
- A5112 XL147Target: PI3KSummary: PI3K inhibitor,selective and reversible
- A5449 PIK-93Summary: PI3Kγ/PI4KIIIβ/PI3Kα inhibitor
- A8354 A66Target: PI3KSummary: P110α inhibitor
- A8488 NVP-BGT226Target: PI3K|mTORSummary: PI3K/mTOR inhibitor,selective and novel
- B2176 GSK1059615Target: PI3K|mTORSummary: PI3K and mTOR inhibitor,potent and reversible
- B1047 GDC-0032Target: PI3KSummary: PI3Kα inhibitor
- B5948 PF-4989216Summary: Selective oral PI3K inhibitor