PI3K
PI3K (phosphatidylinositol-4,5-bisphosphate 3-kinase) is a family of enzymes involved in cellular functions such as cell growth, proliferation, differentiation, motility, survival and intracellular trafficking, which in turn are involved in cancer.
- A8499 PF-04691502Target: Akt|PI3K|mTORSummary: PI3K/mTOR (FRAP) inhibitor
- A8505 PKI-402Summary: PI3K inhibitor,selective, reversible and ATP-competitive
- B2172 PP121Target: mTOR|Eph Receptors|VEGFR|PDGFR|Bcr-Abl|Src|DNA-PK|P110|HckSummary: Dual inhibitor of tyrosine and phosphoinositide kinases
- B2176 GSK1059615Target: PI3K|mTORSummary: PI3K and mTOR inhibitor,potent and reversible
- B7198 PI 828Summary: PI 3-Kinase inhibitor
- B4492 HS-173Target: PI3KSummary: novel PI3K inhibitor
- B4991 GNE-317Summary: potent, brain-penetrant PI3K inhibitor
- B5831 Acalisib (GS-9820)Target: PI3KSummary: PI3Kδ inhibitor
- B5948 PF-4989216Summary: Selective oral PI3K inhibitor
- B5950 AZD8186Target: PI3KSummary: Potent and selective inhibitor of PI3Kβ and PI3Kδ