PI3K
PI3K (phosphatidylinositol-4,5-bisphosphate 3-kinase) is a family of enzymes involved in cellular functions such as cell growth, proliferation, differentiation, motility, survival and intracellular trafficking, which in turn are involved in cancer.
- B5246 740 Y-P5 CitationTarget: PI3KSummary: PI 3-kinase activator,cell permeable
- N1841 QuercetinSummary: Antitumor agent
- B1047 GDC-0032Target: PI3KSummary: PI3Kα inhibitor
- B2186 GSK2636771Target: PI3KSummary: PIK3 inhibitor
- A3005 CAL-101 (Idelalisib, GS-1101)2 CitationTarget: PI3KSummary: PI3K inhibitor
- A3015 BKM1201 CitationTarget: PI3KSummary: Inhibitor of pan-Class I PI3K
- A4097 CUDC-907Target: Histone Deacetylases (HDACs)|PI3KSummary: Potent PI3K/HDAC inhibitor
- A3238 BEZ235 Tosylate1 CitationSummary: MTOR/P13K inhibitor
- A3268 CAL-130 HydrochlorideSummary: PI3K inhibitor
- A3340 CZC24832Summary: Selective PI3K-γ inhibitor