PI3K
PI3K (phosphatidylinositol-4,5-bisphosphate 3-kinase) is a family of enzymes involved in cellular functions such as cell growth, proliferation, differentiation, motility, survival and intracellular trafficking, which in turn are involved in cancer.
- N1841 QuercetinSummary: Antitumor agent
- A3005 CAL-101 (Idelalisib, GS-1101)2 CitationTarget: PI3KSummary: PI3K inhibitor
- A3238 BEZ235 Tosylate1 CitationSummary: MTOR/P13K inhibitor
- A3268 CAL-130 HydrochlorideSummary: PI3K inhibitor
- A3724 PI-103 Hydrochloride1 CitationTarget: PI3K|mTOR|DNA-PKSummary: DNA-PK/PI 3-kinase/mTOR inhibitor
- A2067 PI-1031 CitationSummary: Class I PI3K, mTOR and DNA-PK inhibitor
- A2754 TG100-115Target: PI3KSummary: PI3Kγ/PI3Kδ inhibitor
- A2764 PIK-90Summary: PI3K inhibitor,potent selective
- A1720 Duvelisib (IPI-145, INK1197)Target: PI3KSummary: PI3K-δ/PI3K-γ inhibitor
- B2186 GSK2636771Target: PI3KSummary: PIK3 inhibitor