PI3K
PI3K (phosphatidylinositol-4,5-bisphosphate 3-kinase) is a family of enzymes involved in cellular functions such as cell growth, proliferation, differentiation, motility, survival and intracellular trafficking, which in turn are involved in cancer.
- A3268 CAL-130 HydrochlorideSummary: PI3K inhibitor
- A3340 CZC24832Summary: Selective PI3K-γ inhibitor
- A3432 GDC-0941 dimethanesulfonateSummary: PI3K inhibitor
- A3674 NVP-BKM120 HydrochlorideSummary: PI3K inhibitor
- A3724 PI-103 Hydrochloride1 CitationTarget: PI3K|mTOR|DNA-PKSummary: DNA-PK/PI 3-kinase/mTOR inhibitor
- A3927 VS-5584 (SB2343)Target: PI3K|mTORSummary: MTOR/P13K inhibitor,potent and selective
- A8250 LY 29400263 CitationTarget: PI3KSummary: Potent PI3K inhibitor
- A2067 PI-1031 CitationSummary: Class I PI3K, mTOR and DNA-PK inhibitor
- A2754 TG100-115Target: PI3KSummary: PI3Kγ/PI3Kδ inhibitor
- A5176 AS-605240Target: PI3KSummary: Potent and selective PI 3-Kγ inhibitor