EGFR
EGFR (epidermal growth factor receptor) is the cell-surface receptor of its specific ligands, including epidermal growth factor and TGFα (transforming growth factor α) and is a receptor tyrosine kinase.
- B6377 AG 555Summary: Potent EGFR-kinase inhibitor
- B6378 AG 494Summary: Potent EGFR-kinase inhibitor
- B6989 GW 583340 dihydrochlorideSummary: dual EGFR/ErbB2 tyrosine kinase inhibitor
- B7048 BIBU 1361 dihydrochlorideSummary: EGFR inhibitor
- B7130 PD 158780Summary: ErbB receptor family tyrosine kinase inhibitor
- B7379 JNJ 28871063 hydrochlorideSummary: ErbB receptor family inhibitor
- B7384 CGP 52411Summary: EGFR inhibitor
- A8197 Compound 561 CitationTarget: EGFRSummary: REGFR inhibitor
- A8199 PD153035 hydrochloride1 CitationTarget: EGFRSummary: Potent EGFR inhibitor
- A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: Multitargeted HDAC inhibitor