EGFR
EGFR (epidermal growth factor receptor) is the cell-surface receptor of its specific ligands, including epidermal growth factor and TGFα (transforming growth factor α) and is a receptor tyrosine kinase.
- A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: Multitargeted HDAC inhibitor
- A4139 AG-4903 CitationTarget: EGFR|JAKSummary: JAK2/EGFR inhibitor
- A3240 BIBX 1382Summary: EGFR inhibitor,potent and selective
- A3256 BMS-690514Summary: HER/EGFR inhibitor
- A3320 CO-1686 (AVL-301)1 CitationTarget: EGFRSummary: EGFR inhibitor
- A3397 Erlotinib4 CitationSummary: EGFR tyrosine kinase inhibitor
- A3433 Gefitinib hydrochlorideTarget: EGFRSummary: Potent EGFR inhibitor
- A3482 Icotinib HydrochlorideSummary: EGFR inhibitor,potent and specific
- A3513 IxabepiloneSummary: Epothilone B analog;microtubule-stabilizing agent