MEK1/2
MEK1/2, also known as MAPKK (mitogen-activated protein kinase kinase), is a kinase enzyme which phosphorylates MAPK (mitogen-activated protein kinase).
- A8374 AZD8330Target: MEKSummary: MEK 1/2 inhibitor
- B3261 RO4987655Summary: MEK inhibitor
- B1621 TAK-733Target: MEKSummary: MEK allosteric site inhibitor
- B5727 PD 334581Summary: MEK1 inhibitor
- A9907 MEK Inhibitor SetSummary: For phosphorylation and dephosphorylation applications
- B5817 GDC-09942 CitationSummary: ERK1/2 inhibitor
- B5820 RO5126766(CH5126766)Summary: Raf/MEK dual inhibitor
- B5867 SCH772984 TFASummary: ERK1/2 inhibitor
- B5866 SCH772984 HClSummary: ERK1/2 inhibitor
- B6014 BI-847325Summary: dual inhibitor of MEK and Aurora kinases