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Home >> Signaling Pathways >> GPCR/G protein

GPCR/G protein

  1. Cat.No. Product Name Information
  2. B4876 K-Ras(G12C) inhibitor 12 allosteric inhibitor of K-Ras(G12C)
  3. A8886 UNBS 5162 A pan-antagonist of CXCL chemokines
  4. B7463 RF 9 neuropeptide FF receptors antagonist
  5. B5212 Neuropeptide SF (human) Endogenous antiopiate neuropeptide
  6. B5238 Neuropeptide AF (human) Endogenous antiopioid peptide implicated in pain modulation and endocrine functions
  7. B5386 Neuropeptide FF agonist at NPFF1 and NPFF2 receptors
  8. B5465 Neuropeptide SF (mouse, rat) neuropeptide FF receptor agonist
  9. B5683 RFRP 3 (human) NPFF1 receptor agonist
  10. B6888 N-Formyl-Met-Leu-Phe formyl peptide receptor 1 (FPR1) agonist
  11. B5178 WKYMVM Selective agonist for the formyl peptide receptors FPR2 and FPR3
  12. B5179 WKYMVm Selective agonist for the formyl peptide receptors FPR1, FPR2
  13. B5283 WRW4 Selective antagonist of formyl peptide receptor 2 (FPR2) signaling
  14. B5400 Ac9-25 formyl peptide receptor 1 (FPR1) ligand
  15. B5446 MMK 1 human formyl peptide receptor FPR2 agonist
  16. B5472 Boc-MLF formyl peptide receptor 1 (FPR1) antagonist
  17. B5656 PBP 10 formyl peptide receptor 2 (FPR2) antagonist
  18. B7202 FPR A14 Formyl peptide receptor (FPR) agonist
  19. B5921 Cyclosporin H Selective and competitive formyl peptide receptor antagonist
  20. A3144 Adoprazine 5-HT1A receptor agonist and full D2/3 receptor antagonist
  21. A3159 Alosetron Hydrochloride 5-HT3 receptor antagonist,potent and highly selective
  22. A3192 Asenapine hydrochloride Atypical antipsychotic
  23. A3241 Bilobalide Neuroprotective agent
  24. A3317 Clozapine N-oxide (CNO) Metabolite of clozapine, used in chemogenetics.
  25. A3331 CP-809101 hydrochloride 5-HT2C receptor agonist, potent and selective
  26. A3560 Lu AE58054 5-HT(6)R antagonist
  27. A3561 Lu AE58054 Hydrochloride 5-HT(6)R antagonist
  28. A3748 rac-Rotigotine Hydrochloride Agonist of dopamine D2/D3 receptor
  29. A3776 Rotigotine Agonist of dopamine D2/D3 receptor
  30. A3777 Rotigotine hydrochloride Agonist of dopamine D2/D3 receptor
  31. A3793 SB 271046 hydrochloride Selective 5-HT6 antagonist
  32. A3811 SEA0400 Specific inhibitor of Na+/Ca2+ exchange
  33. A3873 Tianeptine 5-HT facilitator
  34. A3918 Vilazodone Combined SSRI and 5-HT1A receptor partial agonist
  35. A3919 Vilazodone Hydrochloride Combined SSRI and 5-HT1A receptor partial agonist
  36. A3926 Vortioxetine 5-HT receptors antagonist
  37. A3934 WAY-100635 maleate salt 5-hydroxytryptamine 1A antagonist
  38. A1295 Granisetron HCl 5-HT3 receptor antagonist
  39. A1334 Mosapride Citrate 5-HT receptor agonist
  40. A5010 Asenapine Inhibits adrenergic receptor/5-HT receptor
  41. A2436 Fluoxetine HCl Serotonin reuptake inhibitor,selective
  42. A2553 Fluvoxamine maleate Serotonin reuptake inhibitor,selective,antidepressant
  43. A5355 Venlafaxine Dual serotonin/noradrenalin re-uptake inhibitor
  44. A5322 Tianeptine sodium 5-HT uptake facilitator,selective,antidepressant
  45. A5294 Sumatriptan Succinate 5-HT1 receptor agonist
  46. A5350 Ziprasidone HCl Serotonin and dopamine receptor antagonist
  47. A5399 Iloperidone Dopamine (D2) and serotonin (5HT2) receptor antagonist
  48. A2547 Vortioxetine (Lu AA21004) HBr 5-HT receptor modulator, antidepressant and anxiolytic
  49. A2098 PRX-08066 Maleic acid 5-HT2B receptor antagonist,potent and selective
  50. A8514 Risperidone SR-2A inhibitor
  51. A8516 Rizatriptan Benzoate 5-HT Receptor agonist
  52. A8384 Blonanserin Atypical antipsychotic
  53. A8421 Duloxetine HCl 5-HT receptor inhibitor
  54. B1196 Risperidone hydrochloride 5-HT2 receptor blocker
  55. B1197 Risperidone mesylate 5-HT2 receptor blocker
  56. B2265 BRL-15572 5-HT1D receptor antagonist
  57. B2245 BRL-54443 5-HT1E/1F receptor agonist,potent and selective
  58. B1198 Cisapride 5-HT4 receptor agonist
  59. B2256 SB742457 5-HT6 receptor antagonist,highly selective and high affinity
  60. B2240 Olanzapine Antagonist of 5-HT2A and dopamine D2 receptors
  61. B1199 Tandospirone Anxiolytic and antidepressant reagent
  62. B1058 Lasmiditan 5-HT1F receptor agonist
  63. B2254 SB269970 HCl 5-HT7 receptor antagonist,potent and selective
  64. B1200 PRX-08066 5-HT2BR antagonist
  65. B2262 Agomelatine MT1/MT2 / 5-HT2C agonist
  66. B1201 Agomelatine hydrochloride Norepinephrine-dopamine disinhibitor (NDDI)
  67. B1202 Agomelatine L(+)-Tartaric acid Norepinephrine-dopamine disinhibitor (NDDI)
  68. B1001 Loxapine 5-HT receptor antagonist
  69. B1203 Iloperidone hydrochloride D(2)/5-HT(2) receptor antagonistis
  70. B2237 Eletriptan HBr selective 5-HT1B and 5-HT1D receptor agonist
  71. B2229 Palonosetron HCl 5-HT receptor antagonist
  72. B1754 Fenspiride HCl α adrenergic and H1 histamine receptor antagonist
  73. B1204 Ondansetron hydrochloride dihydrate 5-HT3 receptor antagonist
  74. B1002 Tropisetron Hydrochloride 5-HT3 receptor antagonist
  75. B1477 Lurasidone HCl Dopamine D2/5-HT2A/5-HT7/5-HT1A inhibitor
  76. B2258 Tropisetron 5-HT3 receptor antagonist
  77. B1205 Fluvoxamine Selective serotonin reuptake inhibitor
  78. B1206 Pizotifen Highly selective 5-HT receptor blocking agent
  79. B2007 Pizotifen Malate 5-HT receptor antagonist
  80. B1059 Mosapride Selective 5HT4 agonist
  81. B2251 Naratriptan selective 5-HT1 receptor subtype agonist
  82. B2261 Zolmitriptan Potent 5-HT1B/1D/1F agonist
  83. B2231 Amitriptyline HCl Serotonin /norepinephrine receptor/5-HT4/5-HT2 inhibitor
  84. B2263 BMY 7378 5-HT1A partial agonist and α1D adrenoceptor antagonist
  85. B2236 Desvenlafaxine serotonin (5-HT) and norepinephrine (NE) reuptake inhibitor
  86. B2246 Desvenlafaxine Succinate serotonin (5-HT) transporter and norepinephrine (NE) transporter reuptake inhibitor
  87. B2250 LY310762 5-HT1D receptor antagonist
  88. B2253 Prucalopride 5-HT4A and 5-HT4B receptor agonist
  89. B2255 SB271046 5-HT6 receptor antagonist, orally active
  90. B2259 VUF 10166 5-HT3 receptor antagonist
  91. B2260 WAY-100635 Maleate 5-HT1A receptor agonist
  92. B2233 Azasetron HCl 5-HT3 receptor antagonist
  93. B2243 Almotriptan Malate 5-HT1B/1D-receptor agonist
  94. B2241 Ondansetron serotonin 5-HT3 receptor antagonist
  95. B2230 Trazodone HCl 5-HT receptor antagonist
  96. B2234 Clomipramine HCl SERT/NET dopamine transporter (DAT) blocker
  97. B2242 Urapidil HCl α1-adrenoceptor antagonist and 5-HT1A receptor agonist
  98. B2264 Dapoxetine HCl Selective serotonin reuptake inhibitor
  99. B2248 Ketanserin specific 5-HT2A serotonin receptor antagonist
  100. B6558 CP 93129 dihydrochloride 5-HT1B agonist, potent and highly selective
  101. B6306 m-Chlorophenylbiguanide hydrochloride 5-HT3 receptor agonist
  102. B6353 N-Methylquipazine dimaleate 5-HT3 agonist
  103. B6362 Methiothepin maleate 5-HT antagonist
  104. B6383 Quipazine dimaleate 5-HT3 receptor agonist
  105. B6389 MDL 72222 5-HT3 antagonist
  106. B6528 1-Phenylbiguanide hydrochloride 5-HT3 receptor agonist
  107. B6540 Spiperone hydrochloride 5-HT2A serotonin and selective D2-like dopamine receptor antagonist
  108. B6906 PNU 142633 5-HT1D receptor agonist
  109. B7104 PNU 109291 5-HT1D receptor agonist
  110. B7531 WAY 208466 dihydrochloride 5-HT6 agonist
  111. B5027 m-CPP hydrochloride 5-HT2C/2B receptor agonist/partial agonist
  112. B5105 SB 204070 Potent and selective 5-HT4 receptor antagonist
  113. B6308 5-Carboxamidotryptamine maleate 5-HT1 agonist
  114. B6309 Cinanserin hydrochloride 5-HT2 antagonist
  115. B6334 4F 4PP oxalate 5-HT2A antagonist
  116. B6347 Methylergometrine maleate 5-HT1/5-HT2 receptor antagonist
  117. B6352 α-Methyl-5-hydroxytryptamine maleate 5-HT2B receptor agonist
  118. B6365 Metergoline 5-HT1/5-HT2 antagonist
  119. B6399 3-AQC 5-HT3 antagonist
  120. B6423 RS 23597-190 hydrochloride 5-HT4 receptor antagonist
  121. B6427 2-[1-(4-Piperonyl)piperazinyl]benzothiazole 5-HT4 receptor
  122. B6479 MDL 11,939 5-HT2A receptor antagonist
  123. B6513 MK 212 hydrochloride 5-HT2C receptor agonist
  124. B6535 RS 56812 hydrochloride 5-HT3 partial agonist
  125. B6536 RS 67506 hydrochloride potent and selective 5-HT4 partial agonist
  126. B6545 N-Desmethylclozapine 5-HT2C serotonin receptor antagonist
  127. B6548 RS 16566 dihydrochloride ligand for the (R)-zacopride binding site
  128. B6572 GR 55562 dihydrochloride 5-HT1B (5-HT1Dβ) silent antagonist
  129. B6574 BW 723C86 hydrochloride 5-HT2B agonist
  130. B6632 SR 57227 hydrochloride 5-HT3 receptor agonist
  131. B6641 SB 224289 hydrochloride 5-HT1B receptor antagonist
  132. B6653 SB 216641 hydrochloride h5-HT1B antagonist
  133. B6660 SDZ SER 082 fumarate 5-HT2B/2C receptor antagonist
  134. B6685 CP 94253 hydrochloride 5-HT1B agonist
  135. B6688 GR 113808 5-HT4 receptor antagonist
  136. B6708 SB 204741 5-HT2B receptor antagonist
  137. B6709 SB 228357 5-HT2C/2B receptor antagonist
  138. B6713 SB 221284 5-HT2C/2B receptor antagonist
  139. B6729 NAS-181 rat 5-HT1B receptor antagonist
  140. B6754 GR 127935 hydrochloride 5-HT1B/1D receptor antagonist
  141. B6776 LY 215840 5-HT2/5-HT7 receptor antagonist
  142. B6815 Mesulergine hydrochloride 5-HT2A and 2C receptor antagonist
  143. B6818 GR 125487 sulfamate 5-HT4 receptor antagonist
  144. B6819 SB 206553 hydrochloride 5-HT2B/5-HT2C receptor antagonist
  145. B6842 R-96544 hydrochloride 5-HT2 receptor antagonist
  146. B6858 Zacopride hydrochloride 5-HT3 receptor antagonist and 5-HT4 receptor agonist
  147. B6859 WAY 161503 hydrochloride 5-HT2C receptor agonist
  148. B6863 Altanserin hydrochloride 5-HT2A receptor antagonist
  149. B6878 Ro 60-0175 fumarate 5-HT2 receptor agonist
  150. B6898 Ritanserin long-acting 5-HT2 receptor antagonist
  151. B6900 SB 258585 hydrochloride 5-HT6 receptor antagonist
  152. B6902 AS 19 Potent 5-HT7 agonist
  153. B6932 SDZ 205-557 hydrochloride 5-HT3/5-HT4 receptor antagonist
  154. B6958 WAY 629 hydrochloride 5-HT2C agonist
  155. B6973 PNU 22394 hydrochloride 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist
  156. B7032 EMD 386088 hydrochloride 5-HT6 receptor agonist
  157. B7078 Melperone hydrochloride 5-HT2A/D2 receptor antagonist
  158. B7094 LP 44 5-HT7 receptor agonist
  159. B7117 TCB-2 5-HT2A receptor agonist
  160. B7133 L-703,664 succinate 5-HT1D receptor agonist
  161. B7136 Fananserin 5-HT2A receptor antagonist
  162. B7183 Nefazodone hydrochloride 5-HT2A receptor antagonist
  163. B7216 Ro 04-6790 5-HT6 receptor antagonist
  164. B7221 LP 12 hydrochloride 5-HT7 receptor agonist
  165. B7244 1-Methylpsilocin 5-HT2C agonist,potent and selective
  166. B7266 LY 272015 hydrochloride 5-HT2B receptor antagonist
  167. B7267 LY 334370 hydrochloride 5-HT1F receptor agonist
  168. B7270 CJ 033466 5-HT4 partial agonist
  169. B7308 SB 699551 5-ht5a receptor antagonist
  170. B7309 SB 399885 hydrochloride 5-HT6 antagonist
  171. B7344 NPS ALX Compound 4a dihydrochloride 5-HT6 antagonist
  172. B7366 BGC 20-761 5-HT6 antagonist,selective and high affinity
  173. B7377 LY 393558 Dual 5-HT1B/1D receptor antagonist
  174. B7413 ML 10302 hydrochloride 5-HT4 partial agonist
  175. B7437 Org 12962 hydrochloride 5-HT2C receptor agonist
  176. B7461 Donitriptan hydrochloride 5-HT1B/1D receptors agonist, potent and selective
  177. B7470 SGS 518 oxalate 5-HT6 antagonist
  178. B7497 CP 135807 5-HT1D receptor agonist
  179. B7561 NPEC-caged-serotonin 5-HT receptor agonist
  180. B7563 Zotepine 5-HT2A receptor and dopamine D2 receptor antagonist
  181. B7583 LY 266097 hydrochloride 5-HT2B receptor antagonist
  182. B7605 MDL 100907 5-HT2A receptor antagonist
  183. B7616 EMDT oxalate 5-HT6 agonist
  184. B7650 ST 1936 oxalate 5-HT6 receptor agonist
  185. B7660 BIMU 8 5-HT4 agonist
  186. B7690 Tegaserod maleate Partial agonist of 5-HT4
  187. B7723 R 1485 dihydrochloride 5-HT6 antagonist,selective and high affinity
  188. B7729 DR 4485 hydrochloride 5-HT7 antagonist
  189. B7768 NBOH-2C-CN hydrochloride 5-HT2A agonist
  190. B5008 2-Methyl-5-hydroxytryptamine hydrochloride 5-HT3 agonist
  191. B5018 SB 203186 hydrochloride Potent 5-HT4 receptor antagonist
  192. B5026 GR 46611 5-HT1D receptor agonist
  193. B5041 RS 67333 hydrochloride potent and highly selective 5-HT4 partial agonist
  194. B5042 RS 39604 hydrochloride potent and selective 5-HT4 antagonist
  195. B5046 Methysergide maleate Mixed 5-HT1/5-HT2 receptor antagonist
  196. B5104 SB 200646 hydrochloride 5-HT2C/2B receptor antagonist
  197. B5321 DOI hydrochloride Brain penetrant, mixed 5-HT2A/5-HT2C receptor agonist
  198. B5334 SB 258719 hydrochloride Selective 5-HT7 receptor antagonist
  199. B5348 SB 242084 5-HT2C receptor antagonist
  200. B5444 SB 243213 dihydrochloride Selective 5-HT2C inverse agonist
  201. B5540 MS 245 oxalate 5-HT6 antagonist

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