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Telotristat

In stock
Catalog No.
B3247
TPH inhibitor
Grouped product items
SizePriceStock Qty
5mg
$140.00
In stock
10mg
$260.00
In stock
100mg
$1,400.00
In stock

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Background

Telotristat is the active metabolite of LX1606(Telotristat etiprate), which is an orally bioavailable, small-molecule, tryptophan hydroxylase (TPH) inhibitor with potential antiserotonergic activity.

Chemical Properties

StorageStore at RT
M.Wt546.93
Cas No.1033805-28-5
FormulaC25H22ClF3N6O3
Solubility≥27.35mg/mL in DMSO with ultrasonic
Chemical Name(2S)-2-amino-3-[4-[2-amino-6-[(1R)-1-[4-chloro-2-(3-methylpyrazol-1-yl)phenyl]-2,2,2-trifluoroethoxy]pyrimidin-4-yl]phenyl]propanoic acid
SDFDownload SDF
Canonical SMILESCC1=NN(C=C1)C2=C(C=CC(=C2)Cl)C(C(F)(F)F)OC3=NC(=NC(=C3)C4=CC=C(C=C4)CC(C(=O)O)N)N
Shipping ConditionEvaluation sample solution : ship with blue ice.All other available size: ship with RT , or blue ice upon request
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.

Quality Control