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JTC-801

Catalog No.
A8456
KOR-3 (NOP) receptor antagonist
Grouped product items
SizePriceStock Qty
10mM (in 1mL DMSO)
$60.00
In stock
5mg
$45.00
In stock
10mg
$60.00
In stock
50mg
$211.00
In stock

Tel: +1-832-696-8203

Email: [email protected]

Worldwide Distributors

Background

JTC 801 is a high affinity, selective KOR-3 (NOP) receptor antagonist (Ki = 8.2 nM). Displays approximately 12.5-, 129- and 1055-fold selectivity over human μ-, κ- and δ-opioid receptors respectively.

Chemical Properties

Physical AppearanceA solid
StorageStore at -20°C
M.Wt447.96
Cas No.244218-51-7
FormulaC26H25N3O2·HCl
Solubility≥22.4 mg/mL in DMSO; insoluble in H2O; ≥18.27 mg/mL in EtOH with ultrasonic
Chemical NameN-(4-amino-2-methylquinolin-6-yl)-2-[(4-ethylphenoxy)methyl]benzamide;hydrochloride
SDFDownload SDF
Canonical SMILESCCC1=CC=C(C=C1)OCC2=CC=CC=C2C(=O)NC3=CC4=C(C=C3)N=C(C=C4N)C.Cl
Shipping ConditionShip with blue ice, or upon other requests.
General tipsFor obtaining a higher solubility, please warm the tube at 37°C and shake it in the ultrasonic bath for a while. We do not recommend long-term storage for the solution, please use it up soon.

Quality Control

Quality Control & MSDS

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Chemical structure

JTC-801