JTC-801
Catalog No.
A8456
KOR-3 (NOP) receptor antagonist
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JTC 801 is a high affinity, selective KOR-3 (NOP) receptor antagonist (Ki = 8.2 nM). Displays approximately 12.5-, 129- and 1055-fold selectivity over human μ-, κ- and δ-opioid receptors respectively.
| Physical Appearance | A solid |
| Storage | Store at -20°C |
| M.Wt | 447.96 |
| Cas No. | 244218-51-7 |
| Formula | C26H25N3O2·HCl |
| Solubility | ≥22.4 mg/mL in DMSO; insoluble in H2O; ≥18.27 mg/mL in EtOH with ultrasonic |
| Chemical Name | N-(4-amino-2-methylquinolin-6-yl)-2-[(4-ethylphenoxy)methyl]benzamide;hydrochloride |
| SDF | Download SDF |
| Canonical SMILES | CCC1=CC=C(C=C1)OCC2=CC=CC=C2C(=O)NC3=CC4=C(C=C3)N=C(C=C4N)C.Cl |
| Shipping Condition | Evaluation sample solution: ship with blue ice. All other available sizes: ship with RT, or blue ice upon request. |
| General tips | For obtaining a higher solubility, please warm the tube at 37°C and shake it in the ultrasonic bath for a while. Stock solution can be stored below -20°C for several months. |
Quality Control & MSDS
- View current batch:
-
Purity = 98.00%
- COA (Certificate Of Analysis)
- MSDS (Material Safety Data Sheet)
- Datasheet
Chemical structure
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