TAN-452
Catalog No.
BA5646
TAN-452 is an orally active, selective peripherally acting delta opioid receptor antagonist.
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TAN-452 is an orally active, selectively peripherally acting δ-opioid receptor antagonist with a value of 0.47 nM and a value of 0.21 nM.TAN-452 is an antagonist of both μ-opioid receptors (;=36.56 nM; =9.43 nM) and κ-opioid receptors (;=5.31 nM; =7.18 nM).TAN-452 is a a derivative of Naltrindole, has low brain permeability and attenuates morphine-induced side effects without compromising pain control.
| Physical Appearance | A solid |
| Storage | -20°C |
| M.Wt | 486.56 |
| Cas No. | 892039-23-5 |
| Formula | C29H30N2O5 |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |