Histamine Receptor
Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.
- B7071 Proxyfan oxalateSummary: histamine H3 receptor ligand
- B7076 VUF 5681 dihydrobromideSummary: histamine H3 receptor silent antagonist
- B7077 VUF 8430 dihydrobromideSummary: histamine H4 receptor full agonist
- B7451 A 987306Summary: H4 receptor antagonist,potent and selective
- B7495 A 943931 dihydrochlorideSummary: Antagonist of histamine H4 receptor,potent and selective
- B7567 JNJ 10181457 dihydrochlorideSummary: Histamine H3 receptor antagonist
- B7698 A 331440 dihydrochlorideSummary: H3 receptor antagonist,non-imidazole,high affinity
- B5010 (R)-(-)-α-Methylhistamine dihydrobromide1 CitationSummary: Very potent, high affinity H3 agonist
- B5014 DPPE fumarateSummary: inhibitor of histamine binding at the intracellular histamine (Hlc) site
- B5021 TiotidineSummary: Potent histamine H2-receptor antagonist