Histamine Receptor
Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.
- C4153 Doxepin (hydrochloride)Summary: histamine, serotonin, adrenergic, and muscarinic receptors antagonist
- C4255 DimebolinSummary: antihistamine, orally-available
- C5734 Trimipramine (maleate)Summary: potent antagonist of histamine H1 receptor
- B1570 CiproxifanSummary: Histamine H3-receptor antagonist
- B1028 Ciproxifan maleateSummary: Potent histamine H3 receptor antagonist
- B1547 Cetirizine DiHClTarget: Histamine H1 ReceptorsSummary: H1 receptor inverse agonist
- B1553 Tripelennamine HClSummary: H1-receptor antagonist
- B1569 Bepotastine Besilate1 CitationSummary: Non-sedating, selective antagonist of histamine 1 (H1) receptor
- B1562 Ketotifen FumarateSummary: Histamine H1 receptor antagonist
- B1575 LafutidineSummary: Histamine H2-receptor antagonist