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Histamine Receptor

Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.

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Biochemicals

  1. Cat.No. Product Name Information
  2. B1560 Famotidine Histamine H2-receptor antagonist
  3. B1549 Hydroxyzine 2HCl Hydroxyzine is a histamine H1-receptor antagonist, inhibits binding of [3H]pyrilamine/[3H]desloratadine to human histamine H1 receptor with IC50 of 10 nM/19 nM.
  4. B1561 Histamine 2HCl Histamine is an organic nitrogen compound, acts on target cells in mammalian brain via stimulation of Histamine 1/2.
  5. B1573 Fexofenadine HCl Fexofenadine inhibits histamine H1 receptor with IC50 of 246 nM.
  6. B1571 Desloratadine Desloratadine is a potent antagonist for human histamine H1 receptor with IC50 of 51 nM.
  7. B1548 Cyclizine 2HCl Cyclizine 2HCl is a piperazine derivative with Histamine H1 receptor antagonist activity.
  8. B1558 Clemastine Fumarate Clemastine Fumarate (Clemastine) is a selective histamine H1 receptor antagonist with IC50 of 3 nM.
  9. B1556 Chlorpheniramine Maleate Chlorpheniramine (Chlorpheniramine maleate, Chlorphenamine) is an histamine H1 receptor antagonist with IC50 of 12 nM.
  10. B1546 Buclizine HCl Buclizine HCL is an antihistamine and anticholinergic of the piperazine derivative family.
  11. B1555 Betahistine 2HCl Betahistine is a histamine H3 receptors inhibitor with IC50 of 1.9 μM.
  12. B1574 JNJ-7777120 Histamine H4 receptor antagonist
  13. B1550 Levodropropizine Histamine receptor inhibitor,cough suppressant
  14. B1568 Azelastine HCl Azelastine HCl is a potent, second-generation, selective, histamine antagonist.
  15. B1576 Olopatadine HCl Histamine blocker
  16. B1565 Roxatidine Acetate HCl Roxatidine Acetate HCl is a specific and competitive histamin H2 receptor antagonist.
  17. B1545 Brompheniramine hydrogen maleate Brompheniramine maleate is a histamine H1 receptors antagonist.
  18. B1564 Ranitidine Histamine H2-receptor antagonist
  19. B1557 Cimetidine H2 receptor antagonist
  20. B1566 Rupatadine Fumarate Rupatadine is an inhibitor of PAFR and histamine (H1) receptor with Ki of 550 nM and 102 nM, respectively. Phase 2.
  21. B1563 Pemirolast potassium Pemirolast potassium (BMY 26517) is a histamine H1 antagonist and mast cell stabilizer that acts as an antiallergic agent.
  22. B1552 Nizatidine Nizatidine is a histamine H2 receptor antagonist with IC50 of 0.9 nM, also inhibits AChE with IC50 of 6.7 μM.
  23. B1554 Benztropine mesylate Benztropine is a dopamine transporter (DAT) inhibitor with IC50 of 118 nM.
  24. B1118 Mianserin Mianserin is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant.
  25. A3223 Bavisant Human H3 receptor antagonist
  26. A1796 Mianserin HCl 5-HT2 receptor antagonist
  27. A1450 Lidocaine Anasthetic and class Ib antiarrhythmic agent
  28. A3728 Pitolisant oxalate Nonimidazole inverse agonist
  29. A3727 Pitolisant hydrochloride Nonimidazole inverse agonist
  30. A3726 Pitolisant Nonimidazole inverse agonist
  31. A3315 Clemizole H1 histamine receptor antagonist
  32. A3298 Cetirizine Antihistamine
  33. A3225 Bavisant dihydrochloride hydrate Human H3 receptor antagonist
  34. A3224 Bavisant dihydrochloride Human H3 receptor antagonist
  35. A2960 Loratadine Peripheral HH1R antagonist
  36. B1570 Ciproxifan Histamine H3-receptor antagonist
  37. B1567 Azatadine dimaleate Azatadine dimaleate is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.
  38. B1117 Azatadine Azatadine is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.
  39. B1116 Mizolastine dihydrochloride Histamine H1-receptor antagonist
  40. B1551 Mizolastine Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
  41. B1575 Lafutidine Lafutidine, a newly developed histamine H(2)-receptor antagonist, inhibits gastric acid secretion.
  42. B1562 Ketotifen Fumarate Ketotifen (fumarate) is a second-generation noncompetitive H1-antihistamine and mast cell stabilizer, which is used to prevent asthma attacks.
  43. B1569 Bepotastine Besilate Bepotastine Beslilate (Bepreve) is a histamine H1 receptor anatagonist.
  44. B1553 Tripelennamine HCl H1-receptor antagonist
  45. B1547 Cetirizine DiHCl H1 receptor inverse agonist
  46. B1028 Ciproxifan maleate Ciproxifan is an extremely potent histamine H3 inverse agonist/antagonist.
  47. B7229 Methimepip dihydrobromide New Product
  48. B7077 VUF 8430 dihydrobromide New Product
  49. B7076 VUF 5681 dihydrobromide New Product
  50. B7071 Proxyfan oxalate New Product
  51. B7055 JNJ 10191584 maleate New Product
  52. B7049 GT 2016 New Product
  53. B7026 4-Methylhistamine dihydrochloride H4 receptor agonist
  54. B7017 Immethridine dihydrobromide New Product
  55. B7451 A 987306 H4 receptor antagonist,potent and selective
  56. B7495 A 943931 dihydrochloride Antagonist of histamine H4 receptor,potent and selective
  57. B7567 JNJ 10181457 dihydrochloride New Product
  58. B4863 Decloxizine dihydrochloride
  59. B4843 Decloxizine
  60. B5709 VUF 10460 New Product
  61. B5513 JNJ 5207852 dihydrochloride New Product
  62. B5021 Tiotidine New Product
  63. B5014 DPPE fumarate New Product
  64. B5010 (R)-(-)-α-Methylhistamine dihydrobromide New Product
  65. B7698 A 331440 dihydrochloride H3 receptor antagonist,non-imidazole,high affinity
  66. B6931 ROS 234 dioxalate New Product
  67. B6879 Impentamine dihydrobromide New Product
  68. B7072 2-Pyridylethylamine dihydrochloride New Product
  69. B7044 Conessine New Product
  70. B6979 Carcinine ditrifluoroacetate New Product
  71. B6465 ICI 162,846 New Product
  72. B6417 Aminopotentidine New Product
  73. B6398 trans-Triprolidine hydrochloride New Product
  74. B6396 Mepyramine maleate New Product
  75. B6328 Dimaprit dihydrochloride New Product
  76. B7409 Astemizole anti-histamine compound, potent
  77. B6356 (S)-(+)-α-Methylhistamine dihydrobromide New Product
  78. B6357 Nα-Methylhistamine dihydrochloride New Product
  79. B6581 Zolantidine dimaleate New Product
  80. B6510 Immepip dihydrobromide New Product
  81. B6449 Iodophenpropit dihydrobromide New Product
  82. B6437 Clobenpropit dihydrobromide New Product
  83. B6424 Imetit dihydrobromide New Product
  84. B6400 Amthamine dihydrobromide New Product
  85. B6392 HTMT dimaleate New Product
  86. B6390 Thioperamide New Product
  87. B3434 Hydroxyzine Hydroxyzine is a histamine H1-receptor antagonist.
  88. B3309 Cyproheptadine hydrochloride serotonin and histamine antagonist as well as antimuscarinic reagent
  89. B3518 Alcaftadine
  90. B3524 Bilastine