PKC
PKC (protein kinase C) is a serine/threonine protein kinase that mediates insulin signaling, actin cytoskeleton, cell mobility, apoptosis and tumorigenesis etc.
- B1287 Ro 31-8220Target: PKCSummary: pan-PKC inhibitor
- B2191 Dequalinium ChlorideTarget: PKC|Calcium-Activated Potassium (KCa) ChannelsSummary: anti-tumor agent and PKC inhibitor
- B3709 Midostaurin (PKC412)Target: PKC|PKA|KDR|Flk1|PPK|c-Syk|CDK1/CyclinBSummary: PKC inhibitor
- A1670 Enzastaurin (LY317615)2 CitationTarget: PKCSummary: PKC beta inhibitor,potent and selective
- A8341 Go 6976Target: PKCSummary: PKCα/PKCβ1 inhibitor
- A8342 GF 109203X1 CitationTarget: PKCSummary: Protein kinase C,MLCK,PKG and PKA inhibitor
- A8344 K-252cTarget: PKC|PKASummary: Protein kinase inhibitor
- B6803 Rottlerin1 CitationTarget: PKC|Ca2 /calmodulin-dependent protein kinases (CaMKs)|PRAK|MAPKAP-K2Summary: PKC inhibitor
- A8525 Sotrastaurin (AEB071)Target: PKCSummary: PKC inhibitor
- A3306 Chelerythrine ChlorideTarget: PKCSummary: PKC antagonist