Muscarinic Receptor
Muscarinic receptor is a group of G-protein coupled receptors that binds to acetylcholine and mediates cellular responses, including inhibition of acetylate cyclase, phosphoinositide degradation and regulation of potassium channels. It is involved in the neurological diseases such as Alzheimer's and Parkinson's.
- B6949 DAU 5884 hydrochlorideSummary: muscarinic M3 receptor antagonist
- B7003 AQ-RA 741Summary: M2 antagonist,selective and high affinity
- B7114 Zamifenacin fumarateSummary: M3 muscarinic receptor antagonist
- B7123 Milameline hydrochlorideSummary: Muscarinic receptor agonist
- B7285 VU 10010Summary: allosteric potentiator of M4 acetylcholine receptors
- B7448 VU 0238429Summary: positive allosteric modulator of M5 receptors
- B7487 VU 0255035Summary: muscarinic M1 antagonist
- B7636 VU 0357017 hydrochlorideSummary: Positive allosteric modulator of muscarinic M1 receptors
- A3299 CevimelineSummary: Muscarinic receptor agonist
- A3300 Cevimeline hydrochloride hemihydrateSummary: Agonist of muscarinic receptor (M1/M3)