Muscarinic Receptor
Muscarinic receptor is a group of G-protein coupled receptors that binds to acetylcholine and mediates cellular responses, including inhibition of acetylate cyclase, phosphoinositide degradation and regulation of potassium channels. It is involved in the neurological diseases such as Alzheimer's and Parkinson's.
- B7448 VU 0238429Summary: positive allosteric modulator of M5 receptors
- B7487 VU 0255035Summary: muscarinic M1 antagonist
- B7636 VU 0357017 hydrochlorideSummary: Positive allosteric modulator of muscarinic M1 receptors
- B1609 Aclidinium BromideSummary: LAMAs antagonist
- B1620 Tolterodine tartrateTarget: AChRSummary: Competitive muscarinic receptor antagonist
- B1614 Solifenacin succinateTarget: M3 ReceptorsSummary: Muscarinic receptor antagonist
- B1600 Darifenacin HBrTarget: M3 ReceptorsSummary: Selective M3 muscarinic receptor antagonist
- B1618 Fesoterodine FumarateSummary: Muscarinic AChR receptor antagonist
- A3299 CevimelineSummary: Muscarinic receptor agonist
- A3300 Cevimeline hydrochloride hemihydrateSummary: Agonist of muscarinic receptor (M1/M3)