Muscarinic Receptor
Muscarinic receptor is a group of G-protein coupled receptors that binds to acetylcholine and mediates cellular responses, including inhibition of acetylate cyclase, phosphoinositide degradation and regulation of potassium channels. It is involved in the neurological diseases such as Alzheimer's and Parkinson's.
- B6606 Telenzepine dihydrochlorideTarget: M1 ReceptorsSummary: muscarinic M1 receptor antagonist
- B6697 AF-DX 384Summary: M2/M4 selective antagonist
- B6715 McN-A 343Summary: muscarinic M1 receptor agonist
- B6734 (S)-(+)-Dimethindene maleateSummary: M2 muscarinic receptor antagonist
- B6821 PD 102807Summary: M4 muscarinic receptor antagonist
- B6949 DAU 5884 hydrochlorideSummary: muscarinic M3 receptor antagonist
- B7003 AQ-RA 741Summary: M2 antagonist,selective and high affinity
- B7114 Zamifenacin fumarateSummary: M3 muscarinic receptor antagonist
- B7123 Milameline hydrochlorideSummary: Muscarinic receptor agonist
- B7285 VU 10010Summary: allosteric potentiator of M4 acetylcholine receptors