Estrogen/progestogen Receptor
The estrogen/progestogen receptors are activated by the hormone estrogen/progesterone and regulate the gene transcription.
- B5455 G-14 CitationTarget: GPR30Summary: GPR30 agonist, potent and selective
- B5469 G-153 CitationTarget: GPR30Summary: GPER receptor antagonist
- B5707 G-36Summary: G-36 is a selective GPER antagonist
- B4871 OspemifeneSummary: non-hormonal selective estrogen receptor modulator (SERM)
- B5912 ChlorotrianiseneSummary: Estrogen agonist
- B6126 17-HydroxyprogesteroneSummary: endogenous progestogen as well as chemical intermediate in the biosynthesis of other steroid hormones
- B6136 Chlormadinone acetateSummary: steroidal progestin with additional antiandrogen and antigonadotropic effects
- B6143 Hydroxyprogesterone caproateSummary: synthetic progestational agent
- B6167 4-HydroxytamoxifenSummary: estrogen receptor modulator
- B7821 AZD9496Summary: estrogen receptor inhibitor, orally active