Androgen Receptor
AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.
- B7468 CITCO1 CitationTarget: constitutive androstane receptor (CAR)Summary: A selective constitutive androstane receptor (CAR) agonist
- B7503 Cl-4AS-1Summary: steroidal androgen receptor agonist
- A3003 MDV3100 (Enzalutamide)12 CitationTarget: Androgen ReceptorsSummary: Androgen receptor antagonist
- A4326 TAK-700 (Orteronel)2 CitationTarget: human lyaseSummary: Human 17,20-lyase inhibitor
- A3108 17 alpha-propionateSummary: Androgen antagonist
- A3190 ASC-J9Summary: AR degradation enhancer,antiumor agent
- A3780 RU 58841Summary: Androgen receptor antagonist