Androgen Receptor
AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.
- A8364 ARN-5092 CitationTarget: Androgen ReceptorSummary: Androgen receptor inhibitor
- A8404 Cyproterone AcetateSummary: Androgen receptor antagonist
- A8623 TOK-001Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17 inhibitor and androgen receptor (AR) antagonist
- C3186 RD162Summary: androgen receptor (AR) antagonist
- C3546 HE-3235Summary: androgen receptor antagonist
- C3644 DanazolSummary: weak androgenic effects
- C4317 5α-dihydro-11-keto TestosteroneSummary: androgen receptor agonist
- C4721 2-hydroxy FlutamideSummary: androgen receptor inhibitor
- C4768 GSK2881078Summary: selective androgen receptor modulator (SARM)
- B1505 EpiandrosteroneTarget: Voltage-gated Calcium Channels (CaV)Summary: steroid hormone with weak androgenic activity