Androgen Receptor
AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.
- C3546 HE-3235Summary: androgen receptor antagonist
- C3644 DanazolSummary: weak androgenic effects
- C4317 5α-dihydro-11-keto TestosteroneSummary: androgen receptor agonist
- C4721 2-hydroxy FlutamideSummary: androgen receptor inhibitor
- C4768 GSK2881078Summary: selective androgen receptor modulator (SARM)
- B1505 EpiandrosteroneTarget: Voltage-gated Calcium Channels (CaV)Summary: steroid hormone with weak androgenic activity
- B1506 Estradiol valerateTarget: Estrogen and Related ReceptorsSummary: Estrogen receptor agonist
- B1376 FlutamideSummary: Androgen receptor antagonists
- B1378 Spironolactone1 CitationSummary: Competitive mineralocorticoid (aldosterone) receptor antagonist
- B7536 PF 998425Summary: non-steroidal androgen receptor (AR) antagonist